A novel anti-HIV active integrase inhibitor with a favorable in vitro cytochrome P450 and uridine 5'-diphospho-glucuronosyltransferase metabolism profile. (Q30429621)

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English	A novel anti-HIV active integrase inhibitor with a favorable in vitro cytochrome P450 and uridine 5'-diphospho-glucuronosyltransferase metabolism profile.	scientific article

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29 February 2020

A novel anti-HIV active integrase inhibitor with a favorable in vitro cytochrome P450 and uridine 5'-diphospho-glucuronosyltransferase metabolism profile (English)

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29 February 2020

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29 February 2020

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Sanjay Mishra

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Marie K Mankowski

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Marie K Mankowski

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Roger G Ptak

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Priscilla A Hogan

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Priscilla A Hogan

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29 February 2020

author name string

Julie D Russell

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29 February 2020

Jiayi Wei

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18 April 2013

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29 February 2020

Antiviral Research

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29 February 2020

98

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29 February 2020

3

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29 February 2020

365-372

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29 February 2020

Retroviral integrase proteins and HIV-1 DNA integration

1 reference

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Inhibiting early-stage events in HIV-1 replication by small-molecule targeting of the HIV-1 capsid

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Discovery of a Potent HIV Integrase Inhibitor that Leads to a Prodrug with Significant anti-HIV Activity

1 reference

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In Vitro antiretroviral properties of S/GSK1349572, a next-generation HIV integrase inhibitor

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Drug–drug interactions in the treatment of HIV infection: focus on pharmacokinetic enhancement through CYP3A inhibition

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HIV integrase inhibitors as therapeutic agents in AIDS.

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10.1016/J.ANTIVIRAL.2013.04.005

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29 February 2020

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29 February 2020

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29 February 2020

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