Characterisation of the Novel Mixed Mu-NOP Peptide Ligand Dermorphin-N/OFQ (DeNo). (Q36043728)

11 August 2017

Characterisation of the Novel Mixed Mu-NOP Peptide Ligand Dermorphin-N/OFQ (DeNo). (English)

1 reference

11 August 2017

Vanessa Vezzi

5

0 references

Paola Molinari

Paola Molinari

6

0 references

Davide Malfacini

Davide Malfacini

Lorenzo Di Cesare Mannelli

4

0 references

Lorenzo Di Cesare Mannelli

8

0 references

Carla Ghelardini

9

Carla Ghelardini

1 reference

11 August 2017

Maria Camilla Cerlesi

2

Maria Camilla Cerlesi

1 reference

11 August 2017

Mark F Bird

1

1 reference

11 August 2017

Mark Brown

3

1 reference

11 August 2017

Laura Micheli

7

1 reference

11 August 2017

Remo Guerrini

10

1 reference

11 August 2017

Girolamo Calò

11

1 reference

11 August 2017

David G Lambert

12

1 reference

11 August 2017

language of work or name

English

0 references

publication date

7 June 2016

1 reference

11 August 2017

1 reference

11 August 2017

11

1 reference

11 August 2017

6

1 reference

11 August 2017

e0156897

1 reference

Creative Commons Attribution 4.0 International

11 August 2017

start time

7 June 2016

1 reference

April 2022 Public Data File from Crossref

copyright status

copyrighted

0 references

cites work

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MDAN-21: A Bivalent Opioid Ligand Containing mu-Agonist and Delta-Antagonist Pharmacophores and Its Effects in Rhesus Monkeys

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Discovery of a Potent Analgesic NOP and Opioid Receptor Agonist: Cebranopadol

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Functional plasticity of the N/OFQ-NOP receptor system determines analgesic properties of NOP receptor agonists

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Effects of spinally administered bifunctional nociceptin/orphanin FQ peptide receptor/μ-opioid receptor ligands in mouse models of neuropathic and inflammatory pain

2 October 2017

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2 October 2017

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Opiate-Induced Molecular and Cellular Plasticity of Ventral Tegmental Area and Locus Coeruleus Catecholamine Neurons

2 October 2017

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Roles of μ-opioid receptors and nociceptin/orphanin FQ peptide receptors in buprenorphine-induced physiological responses in primates

2 October 2017

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The first universal opioid ligand, (2S)-2-[(5R,6R,7R,14S)-N-cyclopropylmethyl-4,5-epoxy-6,14-ethano-3-hydroxy-6-methoxymorphinan-7-yl]-3,3-dimethylpentan-2-ol (BU08028): characterization of the in vitro profile and in vivo behavioral effects in mous

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Arrestins differentially regulate histamine- and oxytocin-evoked phospholipase C and mitogen-activated protein kinase signalling in myometrial cells.

2 October 2017

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Improving bioscience research reporting: the ARRIVE guidelines for reporting animal research

2 October 2017

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Long-lasting antinociceptive spinal effects in primates of the novel nociceptin/orphanin FQ receptor agonist UFP-112.

2 October 2017

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Heterodimerization of ORL1 and opioid receptors and its consequences for N-type calcium channel regulation.

2 October 2017

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Antinociceptive effects of nociceptin/orphanin FQ administered intrathecally in monkeys

2 October 2017

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The nociceptin/orphanin FQ receptor: a target with broad therapeutic potential

2 October 2017

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Cellular neuroadaptations to chronic opioids: tolerance, withdrawal and addiction

2 October 2017

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Effects of nociceptin/orphanin FQ receptor (NOP) agonist, Ro64-6198, on reactivity to acute pain in mice: comparison to morphine

2 October 2017

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Opioid-induced tolerance and dependence in mice is modulated by the distance between pharmacophores in a bivalent ligand series

2 October 2017

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Heterodimerization of opioid receptor-like 1 and mu-opioid receptors impairs the potency of micro receptor agonist

2 October 2017

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Mitogen-activated protein kinases in apoptosis regulation

2 October 2017

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A role for heterodimerization of mu and delta opiate receptors in enhancing morphine analgesia

2 October 2017

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Protein measurement with the Folin phenol reagent

2 October 2017

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Heterodimerization of mu and delta opioid receptors: A role in opiate synergy

2 October 2017

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Molecular characterization and functional expression of opioid receptor-like1 receptor.

2 October 2017

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Isolation and structure of the endogenous agonist of opioid receptor-like ORL1 receptor

2 October 2017

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Bidirectional modulatory effect of orphanin FQ on morphine-induced analgesia: antagonism in brain and potentiation in spinal cord of the rat.

2 October 2017

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kappa-Opioid agonists produce antinociception after i.v. and i.c.v. but not intrathecal administration in the rat.

11 July 2018

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Opioid receptor desensitization in NG 108-15 cells. Differential effects of a full and a partial agonist on the opioid-dependent GTPase

11 July 2018

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Development and characterisation of novel fentanyl-delta opioid receptor antagonist based bivalent ligands.

11 July 2018

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A novel and facile synthesis of tetra branched derivatives of nociceptin/orphanin FQ.

23 September 2018

1 reference

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Morphine withdrawal produces ERK-dependent and ERK-independent epigenetic marks in neurons of the nucleus accumbens and lateral septum.

23 September 2018

1 reference

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Chimeric G proteins in fluorimetric calcium assays: experience with opioid receptors

23 September 2018

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Facilitation of μ-opioid receptor activity by preventing δ-opioid receptor-mediated codegradation.

23 September 2018

1 reference

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Pharmacological profile of NOP receptors coupled with calcium signaling via the chimeric protein G alpha qi5.

23 September 2018

1 reference

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Binding of the novel radioligand [(3)H]UFP-101 to recombinant human and native rat nociceptin/orphanin FQ receptors

23 September 2018

1 reference

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Nociceptin receptor impairs recognition memory via interaction with NMDA receptor-dependent mitogen-activated protein kinase/extracellular signal-regulated kinase signaling in the hippocampus

23 September 2018

1 reference

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Functional complementation of high-efficiency resonance energy transfer: a new tool for the study of protein binding interactions in living cells.

23 September 2018

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In vitro pharmacological characterisation of a novel cyclic nociceptin/orphanin FQ analogue c[Cys(7,10)]N/OFQ(1-13)NH (2).

23 September 2018

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SR 16435 [1-(1-(bicyclo[3.3.1]nonan-9-yl)piperidin-4-yl)indolin-2-one], a novel mixed nociceptin/orphanin FQ/mu-opioid receptor partial agonist: analgesic and rewarding properties in mice

23 September 2018

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N- and C-terminal modifications of nociceptin/orphanin FQ generate highly potent NOP receptor ligands

23 September 2018

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Evidence for an exclusive antinociceptive effect of nociceptin/orphanin FQ, an endogenous ligand for the ORL1 receptor, in two animal models of neuropathic pain

23 September 2018

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Chronic catheterization of the spinal subarachnoid space

23 September 2018

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Genetic dissociation of opiate tolerance and physical dependence in delta-opioid receptor-1 and preproenkephalin knock-out mice.

23 September 2018

1 reference

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Dimerization of morphine and orphanin FQ/nociceptin receptors: generation of a novel opioid receptor subtype

23 September 2018

1 reference

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Characterization of nociceptin receptors in the periphery: in vitro and in vivo studies

23 September 2018

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Orphanin FQ: a neuropeptide that activates an opioidlike G protein-coupled receptor.

23 September 2018

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Selective blockage of delta opioid receptors prevents the development of morphine tolerance and dependence in mice

23 September 2018

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Acute and subchronic antinociceptive effects of nociceptin/orphanin FQ receptor agonists infused by intrathecal route in rats

23 September 2018

1 reference

Crossref

https://api.crossref.org/works/10.1371%2FJOURNAL.PONE.0156897

AMINO ACID COMPOSITION AND SEQUENCE OF DERMORPHIN, A NOVEL OPIATE-LIKE PEPTIDE FROM THE SKIN OF PHYLLOMEDUSA SAUVAGEI

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/27272042

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1371/JOURNAL.PONE.0156897

1 reference

11 August 2017

0 references

1 reference

11 August 2017

PubMed publication ID

27272042

1 reference